Regioselective electrophilic borylation of haloarenes

Alessandro Del Grosso, Josue Ayuso Carrillo, Michael J. Ingleson*

*Corresponding author for this work

Research output: Contribution to journalArticlepeer-review

Abstract / Description of output

Haloarenes undergo direct borylation using amine:BCl3:AlCl3 in the ratio of 1:1:2. After esterification the pinacol boronate esters are isolated in good yield with regioselectivity controlled by steric and electronic effects.

Original languageEnglish
Pages (from-to)2878-2881
Number of pages4
JournalChemical Communications
Issue number14
Publication statusPublished - 18 Feb 2015


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